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Alkaloid

p-Synephrine · p-Synephrine (bitter orange extract)

A stimulant compound from bitter orange, flagged by EU regulators for cardiovascular risk.

D
Bevisning grade
Mostly animal

Short answer

p-Synephrine (p-Synephrine (bitter orange extract)) is a alkaloid with evidence grade D, meaning it is primarily supported by animal studies. We track 0 produkter containing p-Synephrine. The top-ranked product scores 0 out of 10 on our composite scale (dose, evidence, price, testing, transparency). Prices range up to $0.00 per månad.

Bevisning grade: D Produkter in database: 0 Kategori: Alkaloid

What it is

p-Synephrine is found naturally in bitter orange (Citrus aurantium). It is structurally similar to ephedrine and used in weight loss and pre-workout supplements.

Why people take it

Stimulant effects on heart rate and blood pressure. EU regulators flagged it for restriction due to cardiovascular concerns, especially when combined with caffeine.

Our verdict

Not a longevity ingredient. EU regulators have prioritized it for restriction in supplements.

Structure & class

p-Synephrine is a protoalkaloid. Binds to beta-3 adrenergic receptors. Sympathomimetic activity weaker than ephedrine but potentiated by caffeine.

Mechanism & clinical data

Meta-analyses show modest weight loss benefit but elevated systolic blood pressure and heart rate. Case reports of cardiovascular adverse events.

Pharmacokinetics

Approximately 2 to 3 hours.

Dose & forms

Trial dose
0 mg
/ day
Range in trials
0 to 0 mg
/ day
Common forms
Bitter orange extract, Capsule

What to watch out for

Cardiovascular risk, especially with caffeine. Banned by several sports organizations.

Where this dose comes from

The trial dose above is our editorial pick from the published human trials for this ingredient. We choose the dose that the best-available studies used on the endpoint most relevant to longevity. The range shows the lowest and highest doses tested in published trials. The landmark studies below are the papers we read to set it. You can click through and check our work.

When new trials publish, our automated sweeps flag them. If a new study materially changes the dose, we update it through editorial review and record the old dose, new dose, and the triggering study in every affected product's recommendation history. The dose is never changed automatically.

Regelverk status

EUPrioritized for Article 8 restriction (HoA 2024)
USDSHEA supplement (FDA adverse event reports)
UKRestricted
CANHP with conditions

Timeline

Regelverk events, evidence grade changes, and key research milestones for p-Synephrine, most recent first. Every entry links to its primär source.

  • 2025-04 Regelverk single source
    EU Court sharpens the bar for botanical health claims
    A Court of Justice of the European Union ruling in april 2025 further tightened the requirements for how botanical ingredients (herbs, plant extracts) can be marketed with health claims in the EU, effectively removing much of the flexibility of the on-hold list.
  • 2024-06 Regelverk confirmed
    EU heads of food safety agencies prioritize p-synephrine for restriction
    The HoA Working Group on Food Supplements identified p-synephrine among 12 substances prioritized for Article 8 restriction due to cardiovascular safety concerns, especially when combined with caffeine.
  • 2024-06 Regelverk confirmed
    EU report identifies 117 supplement substances as potential health risks
    The HoA Working Group on Food Supplements (26 European countries) published its first report evaluating 117 substances used in food supplements. Of these, 65 were assessed as likely novel foods, 6 were already regulated, 34 had insufficient data, and 12 were prioritized for Article 8 restriction under Regulation (EC) No 1925/2006. The 12 priority substances include ashwagandha, curcumin, melatonin, piperine, St. John's wort, coumarin, p-synephrine, maca, holy basil, Melaleuca, black cohosh, and L-tryptophan. The report drew on 1,500 RASFF alerts reviewed between 2017 and mid-2022.
  • 2024 Research milestone
    HoA 2024 (BVL/NVWA, EU)
    26-country EU working group prioritized p-synephrine for Article 8 restriction due to cardiovascular safety concerns at supplement doses.
  • 2006-12 Regelverk confirmed
    EU Health Claims Regulation adopted
    Regulation (EC) No 1924/2006 laid down harmonised rules for nutrition and health claims made on foods, including supplements. Only claims listed in the EU Register of authorised claims can be used. Rejected botanical claims are held in a separate on-hold list.
  • 1997 Regelverk confirmed
    EU introduces the Novel Food Regulation
    Regulation (EC) No 258/97 required any food or food ingredient without a history of consumption in the EU before 15 maj 1997 to be authorised before being placed on the market. This is the framework that captures NMN, spermidine as a supplement ingredient, urolithin A, and many other longevity actives.

Landmark studies

  • HoA 2024 (BVL/NVWA, EU)

    26-country EU working group prioritized p-synephrine for Article 8 restriction due to cardiovascular safety concerns at supplement doses.

    Läs studie →

Found in these produkter

Alla produkter in our catalog that contain p-Synephrine, ranked by our overall score. Ranking is editorial, never paid.

No produkter in our catalog contain this yet.

Redaktionellt guides

Buying guides and comparisons

Neighbouring molecules

Related ingredients

Se alla in Alkaloid →

Molekyler in the same class, plus the actives most often formulated alongside p-Synephrine in our catalogue.

Nothing else in the database sits close enough to this molecule to list.

Frequently asked questions

What is p-Synephrine?

p-Synephrine is found naturally in bitter orange (Citrus aurantium). It is structurally similar to ephedrine and used in weight loss and pre-workout supplements.

What dose of p-Synephrine should I take?

The trial dose in published human studies is 0 mg per dag, with a range of 0 to 0 mg per dag. Always consult a qualified clinician before starting any supplement.

Is p-Synephrine safe?

Cardiovascular risk, especially with caffeine. Banned by several sports organizations.

What is the best p-Synephrine supplement?

We track 0 produkter containing p-Synephrine. The top-ranked product scores 0 out of 10 on our composite scale, which evaluates dose, evidence, price, third-party testing, and transparency. See the comparison table above. Scores are editorial judgments, not a scientific standard.

What is the evidence grade for p-Synephrine?

p-Synephrine has evidence grade D, meaning it is primarily supported by animal studies. Grade A means replicated human RCTs with hard endpoints. Grade B means human RCTs with biomarker outcomes. Grade C means mixed or small human trials. See our evidence grading methodology.

Independently checked

Data verification

Bevisning grade
D
Mostly animal
Research dose
0 mg
Verified n/a
Produkter tracked
0
Uppdaterad continuously
Säkerhet signal
Cardiovascular risk, especially with caffeine. Banned by ...
Verified n/a

Bevisning grades are reviewed when new human RCTs are published. Product counts update automatically as new produkter are added. Dose ranges reflect published trial data, not brand recommendations. Read how we verify.